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  1. Aidhen, I. S. (2020). ‘Bioactive C-Glycosides inspired from Natural Products Towards Therapeutics’ in Tiwari, V. K. (ed.) Carbohydrates in Drug Discovery and Development. Amsterdam, Netherlands: Elsevier, pp. 97- 153. 
  2. Synthesis of Benzyl C-Analogues of Dapagliflozin as Potential SGLT2 Inhibitors Mukkamala, R.; Kumar, R.; Banerjee, S. K.; Aidhen, I. S., Eur. J. Org. Chem., 2020, 1828–1839. 
  3. Novel Chemical Scaffolds to Inhibitthe Neutral Amino Acid TransporterB0AT1 (SLC6A19), a Potential Targetto Treat Metabolic Diseases, Yadav, A; Shah, N.;Tiwari, P. K.; Javed, K.; Cheng, Q.; Aidhen, I. S.; Bröer, S. Front. Pharmacol.2020, 11:140, 1-13. 
  4. Natural and Synthetic Glycosylated Chalcones as Promising Bioactive Compounds, Reddy, M. R.; Aidhen, I. S. J. Indian Chem. Soc. 2020, 97, 109-115. 
  5. Acyl and Benzyl-C-β-D-Glucosides: Synthesis and Biostudies for Glucose-Uptake-Promoting Activity in C2C12 Mytotubes, Reddy, M. R.; Hemaiswarya, S.; Kommidi, H.; Aidhen, I. S.; Doble, M. Eur. J. Org. Chem., 2019, 6053–6070. 
  6. Synthesis of 4-C-_-D-GlucosylatedIsoliquiritigenin and Analogues for Aldose Reductase Inhibition StudiesReddy, M. R., Aidhen, I. S.; Reddy, U. A.; Reddy, G. B.; Ingle, K.; Mukhopadhyay, S., Eur. J. Org. Chem., 2019, 3937–3948. 
  7. Discovery of an IsocoumarinAnalogue that Modulates Neuronal Functions via NeurotrophinReceptor TrkB, Bioorg. Med. Chem. Lett., 2019, 29, 585-590.
  8. Synthesis of Unsymmetrical Linear Diarylheptanoids and their Enantiomers and Antiproliferative Activity Studies Sudarshan, K.; Perumal, G.; Aidhen, I. S.; Doble, M. Eur. J. Org. Chem. 2018, Ahead of Print. DOI:10.1002/ejoc.201801211
  9. Convenient Access to 2-β-D-Glucopyranosylpyridines by Using Bohlmann-Rahtz Heteroannulation Reddy, M. R.; Aidhen, I. S. Eur. J. Org. Chem. 2018, 5744-5753.
  10. Effect of flexible, rigid planar and non-planar donors on the performance of dye-sensitized solar cells Unny, D.; Sivanadanam, J.; Mandal, S.; Aidhen, I. S.; Ramanujam, K. J. Electrochem. Soc. 2018, 165, H845-H860.
  11. Design of Cone-Shaped Hole Transporting Material Organic Structures for Perovskite Solar Cells Applications Sivanadanam, J.; Mandal, S.; Aidhen, I. S.; Ramanujam, K. ChemistrySelect 2018, 3, 8159-8166.
  12. Total Synthesis of Natural Product Piperodione and Its Analogues Tiwari, P. K.; Ballav, H.; Aidhen, I. S. ChemistrySelect 2018, 3, 5975-5980.
  13. Exploring the role of the spacers and acceptors on the triphenylamine-based dyes for dye-sensitized solar cells Sivanadanam, J.; Mukkamala, R.; Mandal, S.; Vedarajan, R.; Matsumi, N.; Aidhen, I. S.; Ramanujam, K. Int. J. Hydrogen Energy 2018, 43, 4691-4705.
  14. Synthesis of C-Analogues of β-Glucogallin and Aldose Reductase Inhibition Studies Reddy, M. R.; Aidhen, I. S.; Shruthi, K.; Reddy, G. B. Eur. J. Org. Chem. 2017, 7283-7294.
  15. α,α-Diarylethylene Glycols as Valuable Precursor for Synthesis of 1,1-Diarylethenes and α,α-Diaryl Acetaldehydes Tiwari, P. K.; Sivaraman, B.; Aidhen, I. S. Eur. J. Org. Chem. 2017, 3594-3605.
  16. Stereoselective total synthesis of Oxylipin from open chain gluco-configured building block Borkar, S. R.; Aidhen, I. S. Carbohydr. Res. 2017, 443-444, 23-28.
  17. Synthesis of threo- and erythro-configured trihydroxy open chain lipophilic ketones as possible anti-mycobacterial agents Borkar, S. R.; Bokolia, N.; Aidhen, I. S.; Khan, I. A. Tetrahedron: Asymmetry 2017, 28, 186-195.
  18. Convenient Synthesis of 3-Glycosylated Isocoumarins Sudarshan, K.; Aidhen, I. S. Eur. J. Org. Chem. 2017, 34-38.
  19. Facile Formation of 5-Acylated-2-hydroxymethyl-furans from Open Chain D-Glucosyl-Alkyl/Aryl Ketones Borkar, S. R.; Aidhen, I. S. ChemistrySelect 2016, 1, 6004-6007.
  20. Inhibition of the enzymes in the leukotriene and prostaglandin pathways in inflammation by 3-aryl isocoumarins Ramanan, M.; Sinha, S.; Sudarshan, K.; Aidhen, I. S.; Doble, M. Eur. J. Med. Chem. 2016, 124, 428-434.
  21. Metal-free bipolar/octupolar organic dyes for DSSC application: A combined experimental and theoretical approach Mandal, S.; Kushwaha, S.; Mukkamala, R.; Siripina, V. K.; Aidhen, I. S.; Rajakumar, B.; Kothandaraman, R. Organic Electronics 2016, 36, 177-184.
  22. New building blocks for convenient access to positional isomers of FTY720 and analogues Borkar, S. R.; Bej, R.; Aidhen, I. S. ARKIVOC 2016, 2, 148-161.
  23. A Weinreb Amide Based Building Block for Convenient Access to β,β-Diarylacroleins: Synthesis of 3-Arylindanones Tiwari, P. K.; Aidhen, I. S. Eur. J. Org. Chem. 2016, 2637-2646.
  24. Some interesting 1H NMR features of ortho substituted N-methoxy-N-methyl benzamides Harikrishna, K.; Balasubramaniam, S.; Rakshit, A.; Aidhen, I. S. Indian J. Chem., Sect B 2015, 54B (1), 77-83.
  25. Enhanced two photon absorption cross section and optical nonlinearity of a quasi-octupolar molecule Namboodiri, C. K. R.; Bongu, S. R.; Bisht, P. B.; Mukkamala, R.; Chandra, B.; Aidhen, I. S.; Kelly, T. J.; Costello, J. T. J. Photochem. Photobiol., B: Chemistry 2016, 314, 60-65.
  26. Synthesis of 3-Arylisocoumarins by Using Acyl Anion Chemistry and Synthesis of Thunberginol A and Cajanolactone A By Sudarshan, K.; Manna, M. K.; Aidhen, I. S. Eur. J. Org. Chem. 2015, 1797-1803.
  27. Acyl-anion chemistry for the synthesis of C-aryl glycosides: synthetic efforts towards C-aryl septanosides Harikrishna, K.; Tiwari, P. K.; Aidhen, I. S. Trends Carbohydr. Res. 2014, 6, 37-46.
  28. A Common Building Block for the Syntheses of Amorfrutin and Cajaninstilbene Acid Libraries toward Efficient Binding with Peroxisome Proliferator-Activated Receptors Aidhen, I. S.; Mukkamala, R.; Weidner, C.; Sauer, S. Org. Lett. 2015, 17, 194-197.
  29. A molecular level understanding of interaction between FTY720 (Fingolimod hydrochloride) and DMPC multilamellar vesicles Swain, J.; Borkar, S. R.; Aidhen, I. S.; Mishra, A. K. RSC Advances 2014, 4, 17347-17353.
  30. Iodine-Promoted Oxidative Conversion of o-Vinyl Diaryl Ketones into o-Acetyl Diaryl Ketones, Synthesis of 1-Methyl-4-arylphthalazines as Analogues of Podophyllotoxin Harikrishna, K.; Mukkamala, R.; Hinkelmann, B.; Sasse, F.; Aidhen, I. S. Eur. J. Org. Chem. 2014, 1066-1075.
  31. A Defunctionalization Concept for the Convenient Synthesis of Bis(5-arylfuran-2-yl)methane Scaffolds Tiwari, P. K.; Mukhopadhyay, T.; Aidhen, I. S. Eur. J. Org. Chem. 2013, 8083-8086.
  32. Weinreb amide based building block for convenient access to vinyl ketones Tiwari, P. K.; Aidhen, I. S. Synlett 2013, 24, 1777-1780.
  33. Study of aqueous phase aggregation of FTY720 (fingolimod hydrochloride) and its effect on DMPC liposomes using fluorescent molecular probes Swain, J.; Mohapatra, M.; Borkar, S. R.; Aidhen, I. S.; Mishra, A. K. PCCP, 2013, 15, 17962-17970.
  34. Convenient synthesis of ophiocerin C Borkar, S. R.; Manjunath, B. N.; Aidhen, I. S. Trends Carbohydr. Res. 2013, 5, 34-38.
  35. Study of the Chemoselectivity of Grignard Reagent Addition to Substrates Containing Both Nitrile and Weinreb Amide Functionalities Harikrishna, K.; Rakshit, A.; Aidhen, I. S. Eur. J. Org. Chem. 2013, 4918-4932.
  36. Synthesis of (+)-Centrolobine and Its Analogues by Using Acyl Anion Chemistry Sudarshan, K.; Aidhen, I. S. Eur. J. Org. Chem. 2013, 2298-2302.
  37. Convenient Access to Acyl-Substituted Bis(styrylbenzenes) Based on Building Blocks Using Julia Olefination and Weinreb Amide Chemistry Mukkamala, R.; Senthilmurugan, A.; Aidhen, I. S. Eur. J. Org. Chem. 2013, 2216-2229.
  38. Solvatochromism, multiphoton fluorescence, and resonance energy transfer in a new octupolar dye-pair Namboodiri, C. K. R.; Bisht, P. B.; Mukkamala, R.; Chandra, B.; Aidhen, I. S. Chem. Phys. 2013, 415, 190-195.
  39. Convenient synthesis of D- and L-xylo-1,2,3,4-alkane tetrols from a D-gluco-configured common building block Borkar, S. R.; Manjunath, B. N.; Balasubramaniam, S.; Aidhen, I. S. Carbohydr. Res. 2012, 358, 23-30.
  40. Convenient strategies for the synthesis of 1,4-phenylene spaced sugars Senthilmurugan, A.; Aidhen, I. S. Carbohydr. Res. 2012, 347, 55-63.
  41. Weinreb amide based building blocks for the synthesis of α- and β-organylseleno aryl ketones Balasubramaniam, S.; Aidhen, I. S. Synlett 2011, 11, 1533-1536.
  42. A new fluorescent probe with stimulated emission and multiphoton absorption properties Akbar Ali, S.; Bisht, P. B.; Senthilmurugan, A.; Aidhen, I. S. Chem. Phys. 2011, 382, 68-73.
  43. Weinreb amide based building blocks for convenient access to 1,1-diarylethenes and isocombretastatin analogues Balasubramaniam, S.; Kommidi, H.; Aidhen, I. S. Tetrahedron Lett. 2011, 52, 2683-2686.
  44. Novel synthetic strategy for biphenyl-spaced sugars towards heparinoid mimetics Annamalai, S.; Aidhen, I. S. Trends Carbohydr. Res. 2011, 3, 33-43.
  45. Weinreb Amide Based Building Blocks for Convenient Access to Analogs of Phenstatin Sivaraman, B.; Aidhen, I. S. Eur. J. Org. Chem. 2010, 4991-5003.
  46. Weinreb amide based synthetic equivalents for convenient access to 4-aryl-1,2,3,4-tetrahydroisoquinolines Kommidi, H.; Balasubramaniam, S.; Aidhen, I. S. Tetrahedron 2010, 66, 3723-3729.
  47. Synthesis of (+)-Varitriol Analogues via Novel and Versatile Building Blocks Based on Julia Olefination Senthilmurugan, A.; Aidhen, I. S. Eur. J. Org. Chem. 2010, 555-564.
  48. 2-O-benzylation in D-gluconamide derivative under basic conditions with complete retention of stereo-integrity: convenient access to 2-O-benzyl-3,4:5,6-di-O-isopropylidene-D-glucitol and other differently protected D-glucitol derivatives Manjunath, B. N.; Harikrishna, K.; Aidhen, I. S.; Varghese, B. J. Carbohydr. Chem. 2009, 28, 264-277.
  49. A new distyrylbenzene derivative with Weinreb amide functionality: An efficient laser dye and nonlinear optical material Kalanoor, Basanth S.; Bisht, Prem B.; Annamalai, S.; Aidhen, I. S. J. Lumin. 2009, 129, 1094-1098.
  50. Synthesis of a stable, storable and differentially protected acyclic precursor of D-amicetose and its conversion to 4-O-benzyl-protected D-amicetose Aidhen, I. S.; Satyamurthi, N. Indian J. Chem., Sect. B 2008, 47B, 1851-1857.
  51. The growing synthetic utility of the Weinreb amide Balasubramaniam, S.; Aidhen, I. S. Synthesis 2008, 23, 3707-3738.
  52. Weinreb amide based new synthetic equivalents for convenient access to immunosuppressive agent FTY720 and analogues Balasubramaniam, S.; Annamalai, S.; Aidhen, I. S. Synlett 2007, 18, 2841-2846.
  53. Attempted methylenation of 1,2:3,4:5,6-tri-O-isopropylidene-D-gluconolactone using benzothiazol-2-yl-methylsulfone under Julia conditions yields an unusual product Manjunath, B. N.; Aidhen, I. S.; Varghese, B. J. Carbohydr. Chem. 2007, 26, 17-25.
  54. Synthetic equivalents based on Weinreb amide functionality for convenient access to monoprotected α-diketones Balasubramaniam, S.; Aidhen, I. S. Synlett 2007, 6, 959-963.
  55. An overview of various approaches for the synthesis of 1,2-dideoxy-β-aryl or heteroaryl-D-ribo-furanose framework Mahalingam, S. M.; Manjunath, B. N.; Aidhen, I. S. Proceedings of the Indian National Science Academy, Part A: Physical Sciences 2005, 71, 267-282.
  56. New reagent for convenient access to the α,β-unsaturated N-methoxy-N-methyl-amide functionality by a synthesis based on the Julia olefination protocol Manjunath, B. N.; Sane, N. P.; Aidhen, I. S. Eur. J. Org. Chem. 2006, 2851-2855.
  57. Efficient and rapid regioselective deprotection of isopropylidene ketals Mahalingam, S. M.; Aidhen, I. S. Zeitschrift fuer Naturforschung, B: Chemical Sciences 2005, 60, 962-966.
  58. Propargyl Bromide as an Excellent α-Bromoacetone Equivalent: Convenient and New Route to α-Aroylacetones Mahalingam, S. M.; Aidhen, I. S. J. Org. Chem. 2006, 71, 349-351.
  59. Towards a synthesis of vigabatrin using glycal chemistry Boga, Sobhana B.; Aidhen, Jaimala S.; Aidhen, I. S. Molecules 2005, 10, 871-883.
  60. Convenient enantiopure synthesis of (2S,3R)-2-O-benzyl-3,4-O-isopropylidene-D-erythritol from D-(+)-glucono-δ-lactone: A potential C4 chiral building block Vijayasaradhi, S.; Beedimane, M. N.; Aidhen, I. S. Synthesis 2005, 13, 2267-2269.
  61. Unambiguous Assignment of the Stereochemistry at the Anomeric Carbon in Methyl-α-D-C-Aryl-glucopyranoside Derivative: A Representative of Products from our New Strategy for 2-Deoxy-C-aryl-glucopyranosides Mahalingam, S.; Vijayasaradhi, S.; Aidhen, I.; Varghese, B. J. Carbohydr. Chem. 2005, 24, 321-325.
  62. Simple and highly convenient two-step practical procedure for the synthesis of optically pure methyl D-erythro-2,3-dihydroxybutanoate Mahalingam, S. M.; Sathyamurthi, N.; Aidhen, I. S. Adv. Synth. Catal. 2005, 347, 715-717.
  63. Consequences of rigidity and conformational locking in a 4,4-dimethyl-1,3-dioxolane ring system during protection of internal diol Vijayasaradhi, S.; Aidhen, I. S.; Varghese, B. Carbohydr. Res. 2003, 338, 2899-2903.
  64. Umpolung Strategy for the Synthesis of 2-Deoxy-C-aryl Glycosides: A Serendipitous, Efficient Route for C-Furanoside Analogues Vijayasaradhi, S.; Aidhen, I. S. Org. Lett. 2002, 4, 1739-1742.
  65. Simple synthetic equivalents for the β-(N,N-disubstituted)ethylamino acyl cation synthon and their applications Selvamurugan, V.; Aidhen, I. S. Synthesis 2001, 15, 2239-2246.
  66. N-Methoxy-N-methyl-3-bromopropionamide: a new three carbon homologating agent for the synthesis of unsymmetrical 1,4-diketones Selvamurugan, V.; Aidhen, I. S. Tetrahedron 2001, 57, 6065-6069.
  67. A novel and convenient approach to 5-aryltetrahydro-2-furanols Selvamurugan, V.; Aidhen, I. S. Journal of Chemical Research, Synopses 2000, 12, 590-592.
  68. Synthesis and application of N-methoxy-N-methyl-2-(phenylsulfonyl)acetamide as a two-carbon homologating agent Satyamurthi, N.; Singh, J.; Aidhen, I. S. Synthesis 2000, 3, 375-382.
  69. The growing synthetic utility of Weinreb’s amide Singh, J.; Satyamurthi, N.; Aidhen, I. S. Journal fuer Praktische Chemie 2000, 342, 340-347.
  70. An efficient synthesis of 4,5-O-isopropylidene-protected L-rhodinose Satyamurthi, N.; Aidhen, I. S. Carbohydr. Lett. 1999, 3, 355-360.
  71. Palladium-catalyzed coupling of stannyl allenes with aryl iodides Aidhen, I. S.; Braslau, R. Synth. Commun. 1994, 24, 789-99.
  72. A novel and versatile synthesis of 1-arylbenzocyclobutenols and 1-arylbenzocyclobutenes Aidhen, I. S.; Narasimhan, N. S. Indian J. Chem., Sect B 1993, 32B, 234-238.
  73. A formal synthesis of steganone Aidhen, I. S.; Narasimhan, N. S. Indian J. Chem., Sect B 1993, 32B, 211-221.
  74. Intramolecular arylation of a soft carbon center using manganese(III) acetate: studies towards the spirostructure of fredericamycin-A Aidhen, I. S.; Narasimhan, N. S. Indian J. Chem., Sect B 1993, 32B, 222-228.
  75. A novel synthesis of benzocyclobutenones Aidhen, I. S.; Ahuja, Jaimala R. Tetrahedron Lett. 1992, 33, 5431-2.
  76. A novel and versatile synthesis of 1-aryl-benzocyclobutenols and 1-aryl benzocyclobutenes Aidhen, I. S.; Narasimhan, N. S. Tetrahedron Lett. 1991, 32, 2171-2.
  77. Radical mediated reactions in organic synthesis Narasimhan, N. S.; Aidhen, I. S.; Sunder, N. M. J. Indian Chem. Soc. 1989, 66, 703-9.
  78. Intramolecular arylation of soft carbon center or enolate using manganese(III) acetate: studies towards spirostructure of fredericamycin A Aidhen, I. S.; Narasimhan, N. S. Tetrahedron Lett. 1989, 30, 5323-4.
  79. Acyl anion equivalents in the synthesis of 2H-pyran-2-ones: an efficient synthesis of anibine Dhavale, D. D.; Aidhen, I. S.; Shafique, M. J. Org. Chem. 1989, 54, 3985-7.
  80. Radical-mediated intramolecular arylation using tributyltin hydride-AIBN. A formal synthesis of steganone Narasimhan, N. S.; Aidhen, I. S. Tetrahedron Lett. 1988, 29, 2987-8.
  1. Synthesis of amorfrutin and cajaninstilbene and their analogs from a common building block Aidhen, I. S.; Mukkamala, R. Indian Pat. Appl. 2015, IN 2013CH05457 A 20150529.
  2. A new dye for application in dye laser and nonlinear optics and as a fluorescence lifetime standard Bisht, Prem B.; Aidhen, I. S. Indian Pat. Appl. 2010, IN 2008CH02643 A 20100507
  3. Process for preparation of (βS,4R)- 2,2-dimethyl-β-benzyloxy-1,3-dioxolane-4-ethanol Aidhen, I. S.; Vijayasaradhi, S. Indian Pat. Appl. 2007, IN 2002MA00543 A 20070511.
  4. One pot conversion of D-erythronolactone to enantiomerically pure alkyl (S)-4-bromo-3-hydroxybutanoate Aidhen, I. S.; Gurjar, M. K.; Mahalingam, S. M. Indian Pat. Appl. 2006, IN 2004DE02174 A 20060818.